From bead to flask: Synthesis of a complex β-amido-amide for probe-development studies

نویسندگان

  • Kevin S Martin
  • Cristian Soldi
  • Kellan N Candee
  • Hiromi I Wettersten
  • Robert H Weiss
  • Jared T Shaw
چکیده

A concise synthesis of benzimidazole-substituted β-amido-amide LLW62 is presented. The original synthesis of compounds related to LLW62 was developed on Rink resin as part of a "one-bead, one-compound" combinatorial approach for on-bead screening purposes. The current synthesis is carried out in solution and is amenable to scale-up for follow-up studies on LLW62 and investigations of related structures. The key step involves the use of a β-amino acid-forming three-component reaction (3CR), the scope of which defines its role in the synthetic strategy.

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عنوان ژورنال:

دوره 9  شماره 

صفحات  -

تاریخ انتشار 2013